Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 8BLP
TargetUrea transporter 1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50: 11nMAssay Description:Inhibition of UT-B in human erythrocytes assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50: 11nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50: 11nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50: 25.1nMAssay Description:Reversible inhibition of mouse UT-B-mediated urea transportMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)