Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 8C7X
TargetSerine/threonine-protein kinase B-raf(Human)
University of Orleans

Curated by ChEMBL
LigandPNGBDBM50633493(CHEMBL5440746)
Affinity DataIC50: 48nMAssay Description:Inhibition of B-RAF V600E mutant (unknown origin) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase B-raf(Human)
University of Orleans

Curated by ChEMBL
LigandPNGBDBM50633493(CHEMBL5440746)
Affinity DataIC50: 56nMAssay Description:Inhibition of wild type B-RAF (unknown origin) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)