Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 8H8J
TargetG-protein coupled receptor 35(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50259889(Lodoxamide)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human GPR35 by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetG-protein coupled receptor 35(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50259889(Lodoxamide)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human GPR35 expressed in HEK293 cells co-expressing Galpha16 assessed as increase in calcium mobilization by Fluo-4 AM dye based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetG-protein coupled receptor 35(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50259889(Lodoxamide)
Affinity DataEC50:  4.00E+3nMAssay Description:Agonist activity at human GPR35 expressed in CHO-K1 cells after 90 mins by beta-arrestin 2 recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)