Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) for PDB: 8HUK
LigandPNGBDBM50244350(CHEMBL4091374)
Affinity DataEC50:  366nMAssay Description:Transactivation of mouse GAL4-fused PPARalpha LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50244350(CHEMBL4091374)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50244350(CHEMBL4091374)
Affinity DataEC50:  1.54E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50244350(CHEMBL4091374)
Affinity DataEC50:  3.06E+3nMAssay Description:Agonist activity at PPARalpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50244350(CHEMBL4091374)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at human PPARalpha transfected in African green monkey COS-7 cells co-transfected with pGL4.35 and pBIND reporter gene plasmid asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)