Affinity DataKd: 0.388nMAssay Description:Binding affinity to human CLK1 assessed as dissociation constantMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 4nMAssay Description:Inhibition of human CLK1 assessed as remaining activity by eurofins-cerep kinase profiler analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human CLK4 assessed as incorporation of 33Pi using [gamma-33P]-ATP measured after 60 mins by microplate scintillation counting based ra...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human CLK4 using MBP and [gamma33P]ATP as substrate incubated for 60 mins by radiometric 33PanQinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of N-terminal GST/His6-fused human full length CLK1 (1 to 484 residues) expressed in Sf9 cells assessed as inhibition of autophosphorylati...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human CLK1 assessed as incorporation of 33Pi using [gamma-33P]-ATP measured after 60 mins by microplate scintillation counting based ra...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human CLK1 using myelin basic protein as substrate measured after 70 mins by ADP-GloTM luminescence proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of human CLK4 assessed as remaining activity by eurofins-cerep kinase profiler analysisMore data for this Ligand-Target Pair
