Affinity DataEC50: 80nMAssay Description:Binding affinity to C-terminal full length human MST3 expressed in permeabilized HEK293T cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Binding affinity to C-terminal full length human MST3 expressed in intact HEK293T cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 115nMAssay Description:Binding affinity to N-terminal 6His-tagged TEV fused MST4 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation co...More data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Binding affinity to C-terminal full length human MST4 expressed in permeabilized HEK293T cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.43E+3nMAssay Description:Binding affinity to C-terminal full length human MST4 expressed in intact HEK293T cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair

3D Structure (crystal)