Affinity DataEC50: 50nMAssay Description:Agonist activity at THR-beta in HEK293T cells incubated for 18 to 24 hrs by EnSpire plate reader analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Agonist activity at full length GST-tagged human THR-beta LBD incubated for 1 hr in presence of fluorescein labeled SRC2-2 peptide by Lanthascreen TR...More data for this Ligand-Target Pair

3D Structure (crystal)