Affinity DataIC50: 182nMAssay Description:Binding affinity to human inactivated voltage-gated Na channel 1.7 expressed in HEK293 cells by patch-clamp techniqueMore data for this Ligand-Target Pair
Affinity DataIC50: 1.82E+5nMAssay Description:Inhibition of human Nav1.7 in inactivated condition by manual patch-clamp assayMore data for this Ligand-Target Pair

3D Structure (crystal)