Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 8UD9
TargetProteasome subunit beta type-5(Human)
Cornell University

US Patent
LigandPNGBDBM50600777(CHEMBL5173314 | US20240043470, Compound 3-20)
Affinity DataIC50: 8.18E+4nMAssay Description:Experiments to determine IC50 values against β5i and β5c for compounds were carried out in 96-well plates. In brief, 1 μL of compound ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2024
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetProteasome subunit beta type-5(Human)
Cornell University

US Patent
LigandPNGBDBM50600777(CHEMBL5173314 | US20240043470, Compound 3-20)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunit using Suc-LLVY-AMC as substrate measured after 1.2 hrs in presence of SDSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)