Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 8VKZ
TargetGlucocorticoid receptor(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 445033BDBM445033(US10668167, Compound 41)
Affinity DataIC50: 2.80nMAssay Description:Small molecules were tested for glucocorticoid receptor (GR) binding using the Polarscreen Glucocorticoid Receptor Assay Kit, Red (ThermoFisher A 158...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2021
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetGlucocorticoid receptor(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 445033BDBM445033(US10668167, Compound 41)
Affinity DataIC50: 3nMAssay Description:Inhibition of glucocorticoid receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlucocorticoid receptor(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 445033BDBM445033(US10668167, Compound 41)
Affinity DataEC50:  3nMAssay Description:Agonist activity at glucocorticoid receptor (unknown origin) expressed in K562 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMedPDB3D3D Structure (crystal)