Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 8XBI
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)