Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 8YKI
TargetFibroblast growth factor receptor 2(Human)
Eisai R&D Management

US Patent
LigandChemical structure of BindingDB Monomer ID 142256BDBM142256(US8933099, 22 | US9951047, Compound (I))
Affinity DataIC50: 5.10nMT: 2°CAssay Description:To a flat bottom 96 well white plate (Sumitomo Bakelite Co., Ltd., MS-8496W), 10 μl of FGFR1 protein (Carna Biosciences, Inc., 08-133) solution ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 1(Human)
Eisai R&D Management

US Patent
LigandChemical structure of BindingDB Monomer ID 142256BDBM142256(US8933099, 22 | US9951047, Compound (I))
Affinity DataIC50: 5.70nMT: 2°CAssay Description:To a flat bottom 96 well white plate (Sumitomo Bakelite Co., Ltd., MS-8496W), 10 μl of FGFR1 protein (Carna Biosciences, Inc., 08-133) solution ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 1(Human)
Eisai R&D Management

US Patent
LigandChemical structure of BindingDB Monomer ID 142256BDBM142256(US8933099, 22 | US9951047, Compound (I))
Affinity DataIC50: 5.80nMT: 2°CAssay Description:In this assay, the inhibitory activity of a test substance against the tyrosine kinase activity of FGFR1 protein is measured.To each well of a flat b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2015
Entry Details
US Patent
PDB3D3D Structure (crystal)