Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 9B1G
TargetSolute carrier family 22 member 12(Human)
Fuji Yakuhin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50561689BDBM50561689(Dotinurad | Fyu-981)
Affinity DataIC50: 37nMAssay Description:Inhibition of human URAT1 expressed in Xenopus laevis oocytes assessed as inhibition of [14C]uric acid uptake measured after 60 mins by liquid scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 12(Human)
Fuji Yakuhin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50561689BDBM50561689(Dotinurad | Fyu-981)
Affinity DataIC50: 40nMAssay Description:Inhibition of URAT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 12(Human)
Fuji Yakuhin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50561689BDBM50561689(Dotinurad | Fyu-981)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of URAT1 in human RPTEC assessed as inhibition of [14C]uric acid uptake preincubated for 15 mins followed by [14C]uric acid addition and i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)