Affinity DataIC50: 55nMAssay Description:Antagonist activity at human P2X3R expressed in HEK293 cells incubated for 18 hrs by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair
Affinity DataEC50: 362nMAssay Description:Antagonist activity at alpha, beta-meATP activated human P2X3 receptor by Fluo-4 dye based microplate reader assayMore data for this Ligand-Target Pair

3D Structure (crystal)