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Found 21 Enz. Inhib. hit(s) with all data for entry = 50009688
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  2nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  2nMAssay Description:Inhibition of Platelet glycoprotein IIb/Platelet glycoprotein IIIa binding in unactivated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50055896(3-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isoxa...)
Affinity DataIC50:  4nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50055896(3-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isoxa...)
Affinity DataIC50:  60nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  64nMAssay Description:Inhibition of GPIIb/IIIa binding in activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  64nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  110nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  110nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50055896(3-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isoxa...)
Affinity DataIC50:  112nMAssay Description:Inhibition of GPIIb/IIIa binding in activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50055896(3-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isoxa...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Platelet glycoprotein IIb/Platelet glycoprotein IIIa binding in unactivated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  280nMAssay Description:Inhibition of Platelet glycoprotein IIb/Platelet glycoprotein IIIa binding in unactivated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086631((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086636(1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isoxa...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086633((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086632(1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isoxa...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of GPIIb/IIIa binding in activated human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086634(1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isoxa...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086635((R)-1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-i...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50086630((1-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-isox...)
Affinity DataIC50:  9.80E+6nMAssay Description:Inhibition of platelet aggregation in human platelet rich plasma (hPRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed