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Found 24 Enz. Inhib. hit(s) with all data for entry = 50010022
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090099(5'-Amidinomethyl-17-cyclopropylmethyl-6,7-didehydr...)
Affinity DataKi:  0.214nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090102(5'-N-Biguanidino-17-cyclopropylmethyl-6,7-didehydr...)
Affinity DataKi:  0.226nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090100(CHEMBL319202 | Norbinaltorphimine (norBNI))
Affinity DataKi:  0.244nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090103(5'-(Trimethylammonium)methyl-17-cyclopropylmethyl-...)
Affinity DataKi:  0.354nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090101(5'-Amidino-17-cyclopropylmethyl-6,7-didehydro-4,5a...)
Affinity DataKi:  0.529nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090097(5'-(Dimethylamino)methyl-17-cyclopropylmethyl-6,7-...)
Affinity DataKi:  0.823nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090098(6,7-Dihydro-4,5alpha-epoxy-5'-guanidinyl-17-methyl...)
Affinity DataKi:  2.83nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50068379(5'-[N-(N'-Cyano)guanidinyl]-17-cyclopropylmethyl-6...)
Affinity DataKi:  4.46nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50068379(5'-[N-(N'-Cyano)guanidinyl]-17-cyclopropylmethyl-6...)
Affinity DataKi:  9.46nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090103(5'-(Trimethylammonium)methyl-17-cyclopropylmethyl-...)
Affinity DataKi:  12.8nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090097(5'-(Dimethylamino)methyl-17-cyclopropylmethyl-6,7-...)
Affinity DataKi:  15.7nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090102(5'-N-Biguanidino-17-cyclopropylmethyl-6,7-didehydr...)
Affinity DataKi:  21.5nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090099(5'-Amidinomethyl-17-cyclopropylmethyl-6,7-didehydr...)
Affinity DataKi:  33nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090097(5'-(Dimethylamino)methyl-17-cyclopropylmethyl-6,7-...)
Affinity DataKi:  36nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090099(5'-Amidinomethyl-17-cyclopropylmethyl-6,7-didehydr...)
Affinity DataKi:  40.8nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090100(CHEMBL319202 | Norbinaltorphimine (norBNI))
Affinity DataKi:  41.5nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090100(CHEMBL319202 | Norbinaltorphimine (norBNI))
Affinity DataKi:  49.7nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090101(5'-Amidino-17-cyclopropylmethyl-6,7-didehydro-4,5a...)
Affinity DataKi:  65.7nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090103(5'-(Trimethylammonium)methyl-17-cyclopropylmethyl-...)
Affinity DataKi:  78.4nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50068379(5'-[N-(N'-Cyano)guanidinyl]-17-cyclopropylmethyl-6...)
Affinity DataKi:  89.8nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090102(5'-N-Biguanidino-17-cyclopropylmethyl-6,7-didehydr...)
Affinity DataKi:  108nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090101(5'-Amidino-17-cyclopropylmethyl-6,7-didehydro-4,5a...)
Affinity DataKi:  112nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090098(6,7-Dihydro-4,5alpha-epoxy-5'-guanidinyl-17-methyl...)
Affinity DataKi:  876nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50090098(6,7-Dihydro-4,5alpha-epoxy-5'-guanidinyl-17-methyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity on HEK-293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed