Compile Data Set for Download or QSAR
maximum 50k data
Found 46 Enz. Inhib. hit(s) with all data for entry = 50035359
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124195((R)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  1.5nMAssay Description:In vitro binding affinity to displace [3H]-spiperone from the cloned human dopamine receptor D2 short in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM84637(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Affinity DataKi:  1.80nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM84637(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Affinity DataKi:  24nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM84637(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Affinity DataKi:  52nMAssay Description:Effective concentration for [3H]thymidine uptake in growing CHO cells stably expressing the dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM84637(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Affinity DataKi:  64nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124197((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  120nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124193((S)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  310nMAssay Description:In vitro binding affinity to displace [3H]-spiperone from the cloned human dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124194((R)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  460nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124192((R)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  1.60E+3nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124191((S)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  1.90E+3nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124194((R)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  2.80E+3nMAssay Description:In vitro binding affinity to displace [3H]-spiperone from the cloned human dopamine receptor D2 short in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124194((R)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  2.80E+3nMAssay Description:In vitro binding affinity to displace [3H]-spiperone from the cloned human dopamine receptor D2 short in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124198((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  3.30E+3nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124191((S)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  3.50E+3nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124196((S)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  3.70E+3nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124197((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  4.20E+3nMAssay Description:In vitro binding affinity to displace [3H]-spiperone from the cloned human dopamine receptor D2 short in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124198((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  4.40E+3nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124196((S)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  6.40E+3nMAssay Description:In vitro binding affinity to displace [3H]-spiperone from the cloned human dopamine receptor D2 short in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124192((R)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  7.40E+3nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124196((S)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  8.90E+3nMAssay Description:In vitro Binding affinity towards dopamine D1 receptor using bovine striatal membrane preparations and antagonist [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124191((S)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  9.10E+3nMAssay Description:In vitro Binding affinity towards dopamine D1 receptor using bovine striatal membrane preparations and antagonist [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124197((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  1.00E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124194((R)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  1.20E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124197((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  1.20E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124193((S)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  1.30E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124195((R)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  1.30E+4nMAssay Description:In vitro ability to displace [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124198((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  1.40E+4nMAssay Description:In vitro binding affinity to displace [3H]-spiperone from the cloned human dopamine receptor D2 short in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124192((R)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  1.50E+4nMAssay Description:In vitro Binding affinity towards dopamine D1 receptor using bovine striatal membrane preparations and antagonist [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124191((S)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  1.60E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124191((S)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  1.60E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124196((S)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  1.80E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124194((R)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  1.90E+4nMAssay Description:In vitro Binding affinity towards dopamine D1 receptor using bovine striatal membrane preparations and antagonist [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124198((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  1.90E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124196((S)-2-Phenyl-6-(4-phenyl-piperazin-1-ylmethyl)-5,6...)
Affinity DataKi:  2.00E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124197((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  2.30E+4nMAssay Description:In vitro Binding affinity towards dopamine D1 receptor using bovine striatal membrane preparations and antagonist [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124198((R)-2-Phenyl-5-(4-phenyl-piperazin-1-yl)-4,5,6,7-t...)
Affinity DataKi:  2.30E+4nMAssay Description:In vitro Binding affinity towards dopamine D1 receptor using bovine striatal membrane preparations and antagonist [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124195((R)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  2.50E+4nMAssay Description:In vitro ability to displace [3H]spiperone from the cloned human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124193((S)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  2.90E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124195((R)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  2.90E+4nMAssay Description:In vitro Binding affinity towards dopamine D1 receptor using bovine striatal membrane preparations and antagonist [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124193((S)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  3.00E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 short in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124195((R)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  3.20E+4nMAssay Description:In vitro binding affinity to displace [3H]-spiperone from the cloned human dopamine receptor D2 short in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124193((S)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataKi:  3.90E+4nMAssay Description:In vitro Binding affinity towards dopamine D1 receptor using bovine striatal membrane preparations and antagonist [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124192((R)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  4.30E+4nMAssay Description:In vitro ability to displace [3H]spiperone from the cloned human dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124192((R)-2-(5-Bromo-2-methoxy-phenyl)-4-(4-phenyl-piper...)
Affinity DataKi:  4.40E+4nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50124195((R)-2-Phenyl-4-(4-phenyl-piperazin-1-ylmethyl)-1,4...)
Affinity DataEC50:  50nMAssay Description:Effective concentration for [3H]thymidine uptake in growing CHO cells stably expressing the dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM84637(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Affinity DataEC50:  9.90nMAssay Description:Effective concentration for [3H]thymidine uptake in growing CHO cells stably expressing the dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed