Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50003726
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50162083((5-Methyl-1H-pyrazol-3-yl)-(2-phenyl-quinazolin-4-...)
Affinity DataKi:  24nMAssay Description:Inhibition of Glycogen synthase kinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475257(CHEMBL179420)
Affinity DataKi:  110nMAssay Description:Inhibition of Glycogen synthase kinase-3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475255(CHEMBL179341)
Affinity DataKi:  150nMAssay Description:Inhibition of Glycogen synthase kinase-3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475254(CHEMBL361127)
Affinity DataKi:  250nMAssay Description:Inhibition of Glycogen synthase kinase-3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50033345((5-Methyl-isoxazol-3-yl)-(2-phenyl-quinazolin-4-yl...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of Glycogen synthase kinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475256(CHEMBL176248)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of Glycogen synthase kinase-3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475253(CHEMBL178264)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of Glycogen synthase kinase-3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed