Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50016572
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170869((E)-3-(4'-Hydroxy-biphenyl-4-yl)-acrylic acid | CH...)
Affinity DataEC50: >1.00E+5nMAssay Description:Transcriptional repression in HepG2 cells expressing human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50124518((E)-3-(3'-Adamantan-1-yl-4'-hydroxy-biphenyl-4-yl)...)
Affinity DataEC50:  200nMAssay Description:Binding affinity towards human glucocorticoid receptor (GR) was determined using [3H]-Dexamethasone as radioligand in SF-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170868((E)-3-(4'-Hydroxy-[1,1';3',1'']terphenyl-4-yl)-acr...)
Affinity DataEC50: >1.00E+5nMAssay Description:Binding affinity towards human glucocorticoid receptor (GR) was determined using [3H]-Dexamethasone as radioligand in SF-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170887((E)-3-(3'-Adamantan-1-yl-4'-hydroxy-biphenyl-4-yl)...)
Affinity DataEC50:  7.70E+3nMAssay Description:Binding affinity towards aldosterone receptor (Mineralocorticoid receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170866((E)-3-(3'-Cyclohexylmethyl-4'-hydroxy-biphenyl-4-y...)
Affinity DataEC50:  5.30E+3nMAssay Description:Transcriptional repression in HepG2 cells expressing human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170872((E)-3-(3'-Adamantan-1-yl-4'-hydroxy-biphenyl-4-yl)...)
Affinity DataEC50:  1.76E+4nMAssay Description:Transcriptional repression in HepG2 cells expressing human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed