Compile Data Set for Download or QSAR
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Found 25 Enz. Inhib. hit(s) with all data for entry = 50037725
TargetDelta-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50266025((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi:  0.0310nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50027229(CHEMBL2375157)
Affinity DataKi:  0.0350nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50272081(2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...)
Affinity DataKi:  0.0420nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50266025((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50272081(2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189920((S)-2-amino-N-((S)-2-(2-(benzylamino)-2-oxoethyl)-...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50027229(CHEMBL2375157)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  0.690nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189921(CHEMBL377392 | H-Dmt-Aba-Gly-NH-Ph)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189920((S)-2-amino-N-((S)-2-(2-(benzylamino)-2-oxoethyl)-...)
Affinity DataKi:  11nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189918(CHEMBL211543 | H-Dmt-Aba-Gly-NH-CH2-Bid)
Affinity DataKi:  20nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189921(CHEMBL377392 | H-Dmt-Aba-Gly-NH-Ph)
Affinity DataKi:  27nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189918(CHEMBL211543 | H-Dmt-Aba-Gly-NH-CH2-Bid)
Affinity DataKi:  427nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50027229(CHEMBL2375157)
Affinity DataIC50:  0.130nMAssay Description:Agonist activity at delta opioid receptor by mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50272081(2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...)
Affinity DataIC50:  2.60nMAssay Description:Agonist activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50266025((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataIC50:  2.70nMAssay Description:Agonist activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50272081(2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...)
Affinity DataIC50:  3nMAssay Description:Agonist activity at delta opioid receptor by mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataIC50:  14nMAssay Description:Agonist activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50027229(CHEMBL2375157)
Affinity DataIC50:  27nMAssay Description:Agonist activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189920((S)-2-amino-N-((S)-2-(2-(benzylamino)-2-oxoethyl)-...)
Affinity DataIC50:  51nMAssay Description:Agonist activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189921(CHEMBL377392 | H-Dmt-Aba-Gly-NH-Ph)
Affinity DataIC50:  95nMAssay Description:Agonist activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189918(CHEMBL211543 | H-Dmt-Aba-Gly-NH-CH2-Bid)
Affinity DataIC50:  231nMAssay Description:Agonist activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189921(CHEMBL377392 | H-Dmt-Aba-Gly-NH-Ph)
Affinity DataIC50:  650nMAssay Description:Agonist activity at delta opioid receptor by mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189920((S)-2-amino-N-((S)-2-(2-(benzylamino)-2-oxoethyl)-...)
Affinity DataIC50:  830nMAssay Description:Agonist activity at delta opioid receptor by mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50189918(CHEMBL211543 | H-Dmt-Aba-Gly-NH-CH2-Bid)
Affinity DataIC50:  2.70E+3nMAssay Description:Agonist activity at delta opioid receptor by mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed