Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]diprenorphine from delta opioid receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 144nMAssay Description:Displacement of [3H]diprenorphine from mu opioid receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 153nMAssay Description:Displacement of [3H]diprenorphine from kappa opioid receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum longitudinal muscleMore data for this Ligand-Target Pair
Affinity DataIC50: 215nMAssay Description:Ratio of IC50 of drug to naltrindole for delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair