Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50003835
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50476388(CHEMBL2113281)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]diprenorphine from delta opioid receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50476388(CHEMBL2113281)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]diprenorphine from mu opioid receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50476388(CHEMBL2113281)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]diprenorphine from kappa opioid receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50476388(CHEMBL2113281)
Affinity DataIC50:  0.460nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50476388(CHEMBL2113281)
Affinity DataIC50:  20nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50476388(CHEMBL2113281)
Affinity DataIC50:  215nMAssay Description:Ratio of IC50 of drug to naltrindole for delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed