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Found 15 Enz. Inhib. hit(s) with all data for entry = 50020879
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32783(2-thiophenecarboxylic acid [5-amino-1-(4-fluorophe...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM35509(2-thiophenecarboxylic acid [5-amino-1-(4-methoxyph...)
Affinity DataIC50:  690nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human liver cathepsin B preincubated for 17 hrs in buffer without DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32756(2-furancarboxylic acid [5-amino-1-(4-fluorophenyl)...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human liver cathepsin B preincubated for 2 hrs in buffer without DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human liver cathepsin B preincubated for 2 hrs in non-buffer solution without DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32665(2-furancarboxylic acid [5-amino-1-(4-methylphenyl)...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human liver cathepsin B preincubated for 17 hrs in non-buffer solution without DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32755(2-thiophenecarboxylic acid [5-amino-1-(4-methylphe...)
Affinity DataIC50:  1.99E+3nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human liver cathepsin B preincubated for 24 hrs in buffer without DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human liver cathepsin B preincubated for 24 hrs in non-buffer solution without DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human liver cathepsin B preincubated for 2 hrs in assay buffer with DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50:  4.54E+4nMAssay Description:Inhibition of human liver cathepsin B preincubated for 17 hrs in assay buffer with DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM32784(2-thiophenecarboxylic acid [5-amino-1-(benzenesulf...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human liver cathepsin B preincubated for 24 hrs in assay buffer with DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed