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Found 26 Enz. Inhib. hit(s) with all data for entry = 50038299
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50101075((2S,3S)-3-(3,4-Dichloro-phenyl)-2-methoxycarbonyl-...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50197471((2R,3S)-methyl 3-(3,4-dichlorophenyl)-8-thia-bicyc...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50101075((2S,3S)-3-(3,4-Dichloro-phenyl)-2-methoxycarbonyl-...)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50197471((2R,3S)-methyl 3-(3,4-dichlorophenyl)-8-thia-bicyc...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50197486((2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50197486((2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374510(CHEMBL255140)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374515(CHEMBL399740)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374519(CHEMBL256046)
Affinity DataIC50:  12nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374518(CHEMBL271707)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374516(CHEMBL257482)
Affinity DataIC50:  28nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374515(CHEMBL399740)
Affinity DataIC50:  31nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374518(CHEMBL271707)
Affinity DataIC50:  31nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374510(CHEMBL255140)
Affinity DataIC50:  53nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374512(CHEMBL270659)
Affinity DataIC50:  55nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374516(CHEMBL257482)
Affinity DataIC50:  56nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374513(CHEMBL401554)
Affinity DataIC50:  67nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374519(CHEMBL256046)
Affinity DataIC50:  106nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374514(CHEMBL403660)
Affinity DataIC50:  115nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374514(CHEMBL403660)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374513(CHEMBL401554)
Affinity DataIC50:  405nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374512(CHEMBL270659)
Affinity DataIC50:  593nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374517(CHEMBL407902)
Affinity DataIC50:  992nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374511(CHEMBL279331)
Affinity DataIC50:  1.54E+3nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374511(CHEMBL279331)
Affinity DataIC50:  2.20E+3nMAssay Description:Displacement of [3H]-citalopram from human SERT expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50374517(CHEMBL407902)
Affinity DataIC50:  2.96E+3nMAssay Description:Displacement of [3H]WIN-35428 from human DAT expressed in transfected cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed