Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50026430
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292622(CHEMBL451838 | naphthalen-1-yl 10H-phenothiazine-1...)
Affinity DataKi:  36nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292623(2-tert-butylphenyl 10H-phenothiazine-10-carboxylat...)
Affinity DataKi:  120nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292621(CHEMBL518302 | naphthalen-2-yl 10H-phenothiazine-1...)
Affinity DataKi:  120nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292616(2-methoxyphenyl 10H-phenothiazine-10-carboxylate |...)
Affinity DataKi:  340nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292619(CHEMBL481688 | o-tolyl 10H-phenothiazine-10-carbox...)
Affinity DataKi:  390nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292620(CHEMBL481687 | phenyl 10H-phenothiazine-10-carboxy...)
Affinity DataKi:  570nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292626(3-chlorophenyl 10H-phenothiazine-10-carboxylate | ...)
Affinity DataKi:  570nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292605(2-(diethylamino)ethyl 10H-phenothiazine-10-carboxy...)
Affinity DataKi:  610nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292603(2-(pyrrolidin-1-yl)ethyl 10H-phenothiazine-10-carb...)
Affinity DataKi:  650nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292615(3-methoxyphenyl 10H-phenothiazine-10-carboxylate |...)
Affinity DataKi:  710nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292604(3-(diethylamino)propyl 10H-phenothiazine-10-carbox...)
Affinity DataKi:  740nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292618(CHEMBL481162 | m-tolyl 10H-phenothiazine-10-carbox...)
Affinity DataKi:  1.69E+3nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292624(3-(dimethylamino)phenyl 10H-phenothiazine-10-carbo...)
Affinity DataKi:  1.91E+3nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292614(4-methoxyphenyl 10H-phenothiazine-10-carboxylate |...)
Affinity DataKi:  2.26E+3nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292601(2-morpholinoethyl 10H-phenothiazine-10-carboxylate...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292606(2-(dimethylamino)ethyl 10H-phenothiazine-10-carbox...)
Affinity DataKi:  2.45E+3nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292617(CHEMBL481163 | p-tolyl 10H-phenothiazine-10-carbox...)
Affinity DataKi:  2.85E+3nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292607(CHEMBL520588 | cyclopentyl 10H-phenothiazine-10-ca...)
Affinity DataKi:  3.19E+3nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292602(2-(piperidin-1-yl)ethyl 10H-phenothiazine-10-carbo...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292608(CHEMBL444507 | tert-butyl 10H-phenothiazine-10-car...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292600(CHEMBL480755 | methyl 10H-phenothiazine-10-carboxy...)
Affinity DataKi:  1.02E+4nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292625(4-chlorophenyl 10H-phenothiazine-10-carboxylate | ...)
Affinity DataKi:  1.05E+4nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292609(CHEMBL481142 | butyl 10H-phenothiazine-10-carboxyl...)
Affinity DataKi:  1.34E+4nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292610(CHEMBL450026 | isopropyl 10H-phenothiazine-10-carb...)
Affinity DataKi:  1.81E+4nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292612(CHEMBL481123 | ethyl 10H-phenothiazine-10-carboxyl...)
Affinity DataKi:  2.34E+4nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292613(2-chlorophenyl 10H-phenothiazine-10-carboxylate | ...)
Affinity DataKi:  4.54E+4nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292611(CHEMBL482282 | propyl 10H-phenothiazine-10-carboxy...)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of human serum BchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed