Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) with all data for entry = 50027804
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134030(9-[4-(N,N-dimethylamino)phenylamino]-3,6-bis(3-pyr...)
Affinity DataEC50:  6.30E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP-LIG assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50246816(1,3-Bis(3-(4-(2-(pyrrolidin-1-yl)acetamido)phenylc...)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP-LIG assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50246817(1,3-Bis(3-(4-(3-(pyrrolidin-1-yl)propanamido)pheny...)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP-LIG assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50246818(1,3-Bis(3-(4-(4-(pyrrolidin-1-yl)butanamido)phenyl...)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP-LIG assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50107609(5,10,15,20-tetra(1-methyl-4-pyridyl)-porphyrin | C...)
Affinity DataEC50:  8.90E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP-LIG assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed