Affinity DataKi: >1.90E+3nMAssay Description:Antagonist activity at kappa opioid receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10E+3nMAssay Description:Agonist activity at kappa opioid receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair