Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50038798
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267920((R)-5-(4-Aminophenylamino)-5-oxo-4-(3,4,5-trimetho...)
Affinity DataIC50:  2.34E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267882((R)-5-(4-Fluorophenylamino)-5-oxo-4-(3,4,5-trimeth...)
Affinity DataIC50:  2.43E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267882((R)-5-(4-Fluorophenylamino)-5-oxo-4-(3,4,5-trimeth...)
Affinity DataIC50:  2.61E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267920((R)-5-(4-Aminophenylamino)-5-oxo-4-(3,4,5-trimetho...)
Affinity DataIC50:  3.36E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267918((R)-5-(4-Chlorophenylamino)-5-oxo-4-(3,4,5-trimeth...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267841((R)-5-Oxo-5-4-[(1,3-thiazole-2-amino)sulfonyl]phen...)
Affinity DataIC50:  4.01E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  4.05E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267919((R)-5-(4-Bromophenylamino)-5-oxo-4-(3,4,5-trimetho...)
Affinity DataIC50:  4.19E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267320((R)-5-(4-Chloro-2-fluorobenzylamino)-5-oxo-4-(3,4,...)
Affinity DataIC50:  4.56E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267360((R)-5-(4-Bromo-2-fluorobenzylamino)-5-oxo-4-(3,4,5...)
Affinity DataIC50:  5.12E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267918((R)-5-(4-Chlorophenylamino)-5-oxo-4-(3,4,5-trimeth...)
Affinity DataIC50:  5.23E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267320((R)-5-(4-Chloro-2-fluorobenzylamino)-5-oxo-4-(3,4,...)
Affinity DataIC50:  5.28E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267919((R)-5-(4-Bromophenylamino)-5-oxo-4-(3,4,5-trimetho...)
Affinity DataIC50:  5.44E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267841((R)-5-Oxo-5-4-[(1,3-thiazole-2-amino)sulfonyl]phen...)
Affinity DataIC50:  5.53E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267959((R)-4-(4-Carboxy-2-(3,4,5-trimethoxybenzamido)buta...)
Affinity DataIC50:  5.78E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267958((R)-4-(4-Carboxy-2-(3,4,5-trimethoxybenzamido)buta...)
Affinity DataIC50:  6.58E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267319((R)-5-(3-Iodobenzylamino)-5-oxo-4-(3,4,5-trimethox...)
Affinity DataIC50:  6.59E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267958((R)-4-(4-Carboxy-2-(3,4,5-trimethoxybenzamido)buta...)
Affinity DataIC50:  7.12E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267881((R)-5-(2-Nicotinoylhydrazinyl)-5-oxo-4-(3,4,5-trim...)
Affinity DataIC50:  7.24E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267360((R)-5-(4-Bromo-2-fluorobenzylamino)-5-oxo-4-(3,4,5...)
Affinity DataIC50:  7.61E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267319((R)-5-(3-Iodobenzylamino)-5-oxo-4-(3,4,5-trimethox...)
Affinity DataIC50:  7.68E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267317((R)-5-(3-Chloro-4-fluorophenylamino)-5-oxo-4-(3,4,...)
Affinity DataIC50:  7.85E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267961((R)-5-(2,5-Dichlorophenylamino)-5-oxo-4-(3,4,5-tri...)
Affinity DataIC50:  8.04E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267959((R)-4-(4-Carboxy-2-(3,4,5-trimethoxybenzamido)buta...)
Affinity DataIC50:  8.63E+4nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267880((R)-5-Oxo-5-(2-(thiazole-2-carbonyl)hydrazinyl)-4-...)
Affinity DataIC50:  8.77E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267960((R)-5-(2,4-Difluorophenylamino)-5-oxo-4-(3,4,5-tri...)
Affinity DataIC50:  8.96E+4nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267842((R)-5-[4-(Aminosulfonyl)phenylamino]-5-oxo-4-[(3,4...)
Affinity DataIC50:  1.03E+5nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267432(CHEMBL476466 | N-(1-(2-Aminophenyl)-2,6-dioxopiper...)
Affinity DataIC50:  1.04E+5nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267317((R)-5-(3-Chloro-4-fluorophenylamino)-5-oxo-4-(3,4,...)
Affinity DataIC50:  1.07E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267879((R)-5-Oxo-5-(thiazol-2-ylamino)-4-(3,4,5-trimethox...)
Affinity DataIC50:  1.08E+5nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267960((R)-5-(2,4-Difluorophenylamino)-5-oxo-4-(3,4,5-tri...)
Affinity DataIC50:  1.09E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267881((R)-5-(2-Nicotinoylhydrazinyl)-5-oxo-4-(3,4,5-trim...)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267961((R)-5-(2,5-Dichlorophenylamino)-5-oxo-4-(3,4,5-tri...)
Affinity DataIC50:  1.22E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267880((R)-5-Oxo-5-(2-(thiazole-2-carbonyl)hydrazinyl)-4-...)
Affinity DataIC50:  1.69E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267318((R)-5-(3-Bromobenzylamino)-5-oxo-4-(3,4,5-trimetho...)
Affinity DataIC50:  1.77E+5nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267318((R)-5-(3-Bromobenzylamino)-5-oxo-4-(3,4,5-trimetho...)
Affinity DataIC50:  2.87E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267879((R)-5-Oxo-5-(thiazol-2-ylamino)-4-(3,4,5-trimethox...)
Affinity DataIC50:  3.69E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267433((R)-5-(2-Chloroethylamino)-5-oxo-4-(3,4,5-trimetho...)
Affinity DataIC50:  5.02E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267842((R)-5-[4-(Aminosulfonyl)phenylamino]-5-oxo-4-[(3,4...)
Affinity DataIC50:  6.28E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267432(CHEMBL476466 | N-(1-(2-Aminophenyl)-2,6-dioxopiper...)
Affinity DataIC50:  6.60E+5nMAssay Description:Inhibition of MMP2 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50267433((R)-5-(2-Chloroethylamino)-5-oxo-4-(3,4,5-trimetho...)
Affinity DataIC50:  8.05E+5nMAssay Description:Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed