Compile Data Set for Download or QSAR
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Found 18 Enz. Inhib. hit(s) with all data for entry = 50031432
TargetMu-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313166((S)-(2-hydroxy-6-methylphenyl)(2,3,5,7a-tetrahydro...)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313167((S,E)-(2,3,5,6,7,9a-hexahydro-1H-pyrrolo[1,2-a]aze...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]U69593 from rat kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50211219(elaeocarpenine)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]U69593 from rat kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313167((S,E)-(2,3,5,6,7,9a-hexahydro-1H-pyrrolo[1,2-a]aze...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50211219(elaeocarpenine)
Affinity DataKi:  1.40E+4nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50211219(elaeocarpenine)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313164((S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-metho...)
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]U69593 from rat kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313163((S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-hydro...)
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [3H]U69593 from rat kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313166((S)-(2-hydroxy-6-methylphenyl)(2,3,5,7a-tetrahydro...)
Affinity DataKi:  3.50E+4nMAssay Description:Displacement of [3H]U69593 from rat kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313163((S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-hydro...)
Affinity DataKi:  4.50E+4nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313165((S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-hydro...)
Affinity DataKi:  4.90E+4nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313165((S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-hydro...)
Affinity DataKi:  8.30E+4nMAssay Description:Displacement of [3H]U69593 from rat kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313163((S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-hydro...)
Affinity DataKi:  9.40E+4nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313167((S,E)-(2,3,5,6,7,9a-hexahydro-1H-pyrrolo[1,2-a]aze...)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313165((S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-hydro...)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313166((S)-(2-hydroxy-6-methylphenyl)(2,3,5,7a-tetrahydro...)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313164((S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-metho...)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50313164((S)-(1,2,3,5,6,8a-hexahydroindolizin-8-yl)(2-metho...)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed