Affinity DataKi: 2.00E+3nMAssay Description:Activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant CYP2D6 by spectrafluorometryMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 7.94E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CYP2D6 by spectrafluorometryMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by scintillation proximity assayMore data for this Ligand-Target Pair