Affinity DataKi: 3.20E+3nMAssay Description:Binding affinity to GluR2More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Novartis Pharma
Curated by ChEMBL
Novartis Pharma
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity to GluR5More data for this Ligand-Target Pair
Affinity DataKi: 9.20E+3nMAssay Description:Binding affinity to GluR1More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+4nMAssay Description:Binding affinity to GluR3More data for this Ligand-Target Pair
Affinity DataKi: 5.05E+4nMAssay Description:Binding affinity to GluR4More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Novartis Pharma
Curated by ChEMBL
Novartis Pharma
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to GluR6More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Novartis Pharma
Curated by ChEMBL
Novartis Pharma
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to GluR7More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human OAT1More data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of human OAT3More data for this Ligand-Target Pair