Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50032054
TargetGlutamate receptor 2(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM86751(CHEMBL14935 | LY 293558 | LY-293558)
Affinity DataKi:  3.20E+3nMAssay Description:Binding affinity to GluR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM86751(CHEMBL14935 | LY 293558 | LY-293558)
Affinity DataKi:  4.20E+3nMAssay Description:Binding affinity to GluR5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM86751(CHEMBL14935 | LY 293558 | LY-293558)
Affinity DataKi:  9.20E+3nMAssay Description:Binding affinity to GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM86751(CHEMBL14935 | LY 293558 | LY-293558)
Affinity DataKi:  3.20E+4nMAssay Description:Binding affinity to GluR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM86751(CHEMBL14935 | LY 293558 | LY-293558)
Affinity DataKi:  5.05E+4nMAssay Description:Binding affinity to GluR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM86751(CHEMBL14935 | LY 293558 | LY-293558)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to GluR6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM86751(CHEMBL14935 | LY 293558 | LY-293558)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to GluR7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50133599((7-Imidazol-1-yl-6-nitro-2,3-dioxo-3,4-dihydro-2H-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human OAT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50133599((7-Imidazol-1-yl-6-nitro-2,3-dioxo-3,4-dihydro-2H-...)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of human OAT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed