Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50031824
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50320022((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50320023((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50320024((S)-N-(3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylami...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50320023((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataKi:  7.30E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50320022((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataIC50:  15nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50320022((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataIC50:  25nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50320024((S)-N-(3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylami...)
Affinity DataIC50:  170nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50320023((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataIC50:  330nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50320022((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataIC50:  390nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataIC50:  510nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50320023((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataIC50:  1.10E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50320024((S)-N-(3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylami...)
Affinity DataIC50:  1.90E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed