TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 345nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
Affinity DataKi: 590nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 99nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 104nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 136nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 175nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 740nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.45E+3nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair