Compile Data Set for Download or QSAR
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Found 53 Enz. Inhib. hit(s) with all data for entry = 50032710
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333561(2-{5-Chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahy...)
Affinity DataIC50:  8nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333572(2-{5-Chloro-2-[9-(2-methoxy-acetyl)-6,7,8,9-tetrah...)
Affinity DataIC50:  13nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333567(2-[5-Chloro-2-(9-ethyl-6,7,8,9-tetrahydro-5-oxa-9-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333575(2-[2-(9-Acetyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benz...)
Affinity DataIC50:  17nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333567(2-[5-Chloro-2-(9-ethyl-6,7,8,9-tetrahydro-5-oxa-9-...)
Affinity DataIC50:  18nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333561(2-{5-Chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahy...)
Affinity DataIC50:  19nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333571(2-{5-Chloro-2-[9-(2-pyrrolidin-1-yl-acetyl)-6,7,8,...)
Affinity DataIC50:  19nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333558(2-{5-Chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahy...)
Affinity DataIC50:  20nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333568(2-{5-Chloro-2-[9-(2-pyrrolidin-1-yl-ethyl)-6,7,8,9...)
Affinity DataIC50:  21nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333568(2-{5-Chloro-2-[9-(2-pyrrolidin-1-yl-ethyl)-6,7,8,9...)
Affinity DataIC50:  22nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333559(3-Chloro-2-{5-chloro-2-[3-(2-methoxy-ethyl)-2,3,4,...)
Affinity DataIC50:  24nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333563(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  25nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333560(2-{5-Chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahy...)
Affinity DataIC50:  26nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333570(2-[2-(9-Acetyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benz...)
Affinity DataIC50:  28nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333566(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  28nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333570(2-[2-(9-Acetyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benz...)
Affinity DataIC50:  30nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333562(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  32nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333563(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  36nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333558(2-{5-Chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahy...)
Affinity DataIC50:  41nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333574(2-[5-Chloro-2-(9-ethyl-6,7,8,9-tetrahydro-5-oxa-9-...)
Affinity DataIC50:  41nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333569(2-[5-Chloro-2-(6,7,8,9-tetrahydro-5-oxa-9-aza-benz...)
Affinity DataIC50:  42nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333571(2-{5-Chloro-2-[9-(2-pyrrolidin-1-yl-acetyl)-6,7,8,...)
Affinity DataIC50:  44nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333566(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  45nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333562(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  46nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333564(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  47nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333575(2-[2-(9-Acetyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benz...)
Affinity DataIC50:  49nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333565(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  50nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333572(2-{5-Chloro-2-[9-(2-methoxy-acetyl)-6,7,8,9-tetrah...)
Affinity DataIC50:  51nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333564(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  53nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333569(2-[5-Chloro-2-(6,7,8,9-tetrahydro-5-oxa-9-aza-benz...)
Affinity DataIC50:  57nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333565(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  81nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333574(2-[5-Chloro-2-(9-ethyl-6,7,8,9-tetrahydro-5-oxa-9-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333573(2-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  140nMAssay Description:Inhibition of c-Met cytoplasmic domain expressed in baculovirus after 30 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333558(2-{5-Chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahy...)
Affinity DataIC50:  220nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333561(2-{5-Chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahy...)
Affinity DataIC50:  230nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333568(2-{5-Chloro-2-[9-(2-pyrrolidin-1-yl-ethyl)-6,7,8,9...)
Affinity DataIC50:  300nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333567(2-[5-Chloro-2-(9-ethyl-6,7,8,9-tetrahydro-5-oxa-9-...)
Affinity DataIC50:  370nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333573(2-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  440nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333574(2-[5-Chloro-2-(9-ethyl-6,7,8,9-tetrahydro-5-oxa-9-...)
Affinity DataIC50:  490nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333570(2-[2-(9-Acetyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benz...)
Affinity DataIC50:  500nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333562(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  550nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333559(3-Chloro-2-{5-chloro-2-[3-(2-methoxy-ethyl)-2,3,4,...)
Affinity DataIC50:  550nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333569(2-[5-Chloro-2-(6,7,8,9-tetrahydro-5-oxa-9-aza-benz...)
Affinity DataIC50:  560nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333565(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  800nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333564(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  820nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333572(2-{5-Chloro-2-[9-(2-methoxy-acetyl)-6,7,8,9-tetrah...)
Affinity DataIC50:  930nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333563(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333575(2-[2-(9-Acetyl-6,7,8,9-tetrahydro-5-oxa-9-aza-benz...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333560(2-{5-Chloro-2-[3-(2-methoxy-ethyl)-2,3,4,5-tetrahy...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of c-Met expressed in human GTL-16 cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50333566(3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylam...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of insulin receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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