Compile Data Set for Download or QSAR
maximum 50k data
Found 43 Enz. Inhib. hit(s) with all data for entry = 50033088
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339236((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339240((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339242((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  0.820nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339233((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  0.930nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  1.35nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339238((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50095155((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339237((1R,2S)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339231((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339232((1S,2R)-N-((S)-1-((2R,3R)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  4.11nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339235((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339239((1S,2R)-N-((S)-1-((2R,3R)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339243((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  11.1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339241((1S,2R)-N-((S)-1-((2R,3R)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  33.9nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339234((1S,2R)-N-((S)-1-((2R,3R)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  34.6nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339236((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339233((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  123nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339240((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  142nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339230((1R,2S)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339239((1S,2R)-N-((S)-1-((2R,3R)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  198nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339232((1S,2R)-N-((S)-1-((2R,3R)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  287nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339238((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  366nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339231((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  571nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339242((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  661nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339237((1R,2S)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  689nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339241((1S,2R)-N-((S)-1-((2R,3R)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  1.27E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339235((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  1.44E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339243((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  2.64E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339234((1S,2R)-N-((S)-1-((2R,3R)-1-amino-1-oxo-3-phenylbu...)
Affinity DataKi:  3.36E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50095155((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  4.17E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339230((1R,2S)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataKi:  7.82E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  8.77E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339240((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339238((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataEC50:  92nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339236((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataEC50:  51nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataEC50:  214nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50095155((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataEC50:  166nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339235((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataEC50:  264nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339233((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataEC50:  22.1nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339231((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataEC50:  380nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339242((1S,2R)-N-((S)-1-((2S,3S)-1-amino-1-oxo-3-phenylbu...)
Affinity DataEC50:  273nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataEC50:  212nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50339243((1S,2R)-N-((2S)-1-(1-amino-3-(4-fluorophenyl)-1-ox...)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at mu opioid receptor in rat brain membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed