Compile Data Set for Download or QSAR
maximum 50k data
Found 375 Enz. Inhib. hit(s) with all data for entry = 50033028
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  18nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338432((R)-1-(1-(5-(aminooxycarbonyl)pyridin-3-yl)piperid...)
Affinity DataIC50:  18nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338439(3-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethyl)pipe...)
Affinity DataIC50:  21nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50140533(CHEMBL25211 | N-[4-((S)-1-Amino-2-oxo-2-thiazolidi...)
Affinity DataIC50:  22nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338440(CHEMBL1682974 | trans-N-(4-((S)-1-amino-2-oxo-2-(t...)
Affinity DataIC50:  33nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338458(CHEMBL1683092 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  38nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338438(3-(4-((R)-1-amino-2-(2,5-difluorophenyl)ethyl)pipe...)
Affinity DataIC50:  51nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338437(CHEMBL1683143 | methyl 3-(4-((R)-1-amino-2-(2,5-di...)
Affinity DataIC50:  54nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338457(CHEMBL1683091 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  55nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338413(CHEMBL1683119 | trans-1-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  57nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338415(CHEMBL1683121 | trans-(R)-1-(4-((R)-1-amino-2-(2,5...)
Affinity DataIC50:  70nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338429((R)-2-(2,5-difluorophenyl)-1-(1-(2,6-dimethylpyrid...)
Affinity DataIC50:  71nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338436((R)-5-(4-(1-amino-2-(2,5-difluorophenyl)ethyl)pipe...)
Affinity DataIC50:  72nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338434((R)-2-(2,5-difluorophenyl)-1-(1-(pyrimidin-5-yl)pi...)
Affinity DataIC50:  75nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338428((R)-5-(4-(1-amino-2-(2,5-difluorophenyl)ethyl)pipe...)
Affinity DataIC50:  77nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338435((R)-2-(2,5-difluorophenyl)-1-(1-(2-methoxypyrimidi...)
Affinity DataIC50:  78nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338431((R)-ethyl 5-(4-(1-amino-2-(2,5-difluorophenyl)ethy...)
Affinity DataIC50:  82nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338448(CHEMBL1682982 | trans-4-(N-(4-((R)-1-amino-2-(2,5-...)
Affinity DataIC50:  84nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338443(CHEMBL1682977 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  85nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338451(CHEMBL1682985 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  94nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338447(CHEMBL1682981 | trans-3-(N-(4-((R)-1-amino-2-(2,5-...)
Affinity DataIC50:  99nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338405(CHEMBL1683112 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  100nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338455(CHEMBL1683089 | trans-N-(5-(N-(4-((R)-1-amino-2-(2...)
Affinity DataIC50:  100nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338456(CHEMBL1683090 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338473(CHEMBL1683107 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338467(CHEMBL1683101 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338404(CHEMBL1683111 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338442(CHEMBL1682976 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338430((R)-2-(2,5-difluorophenyl)-1-(1-(6-fluoropyridin-3...)
Affinity DataIC50:  110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338426((R)-2-(2,5-difluorophenyl)-1-(1-(pyridin-3-yl)pipe...)
Affinity DataIC50:  110nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338472(CHEMBL1683106 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  120nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338464(CHEMBL1683098 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  120nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338471(CHEMBL1683105 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  120nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338450(CHEMBL1682984 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  130nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338466(CHEMBL1683100 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  130nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338424((R)-2-(2,5-difluorophenyl)-1-(1-(methylsulfonyl)pi...)
Affinity DataIC50:  130nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338474(CHEMBL1683108 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338475(CHEMBL1683109 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338441(CHEMBL1682975 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338445(CHEMBL1682979 | trans-4-amino-N-(4-((R)-1-amino-2-...)
Affinity DataIC50:  140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338469(CHEMBL1683103 | trans-4-((4-((R)-1-amino-2-(2,5-di...)
Affinity DataIC50:  140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338470(CHEMBL1683104 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  140nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338449(CHEMBL1682983 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  150nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338454(CHEMBL1683088 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  170nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338440(CHEMBL1682974 | trans-N-(4-((S)-1-amino-2-oxo-2-(t...)
Affinity DataIC50:  170nMAssay Description:Inhibition of DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338444(CHEMBL1682978 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  180nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338414(CHEMBL1683120 | trans-(S)-1-(4-((R)-1-amino-2-(2,5...)
Affinity DataIC50:  200nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338420(CHEMBL1683126 | trans-3-(((4-((R)-1-amino-2-(2,5-d...)
Affinity DataIC50:  220nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338461(CHEMBL1683095 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  260nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338476(CHEMBL1683110 | trans-N-(4-((R)-1-amino-2-(2,5-dif...)
Affinity DataIC50:  260nMAssay Description:Inhibition of DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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