TargetKappa-type opioid receptor(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membranes after 150 mins by scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membranes after 150 mins by scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membranes after 150 mins by scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membranes after 150 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 89nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 221nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 221nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 378nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membranes after 150 mins by scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 378nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membranes after 150 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 452nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 531nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: 531nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membranes after 150 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair