Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50033533
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataIC50:  3nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataIC50:  170nMAssay Description:Inhibition of human VPS34More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataIC50:  437nMAssay Description:Inhibition of PI3K C2betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataIC50:  922nMAssay Description:Inhibition of P110alpha/p85alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of PI3K C2alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of P110delta/p85alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of P110gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataIC50:  3.44E+3nMAssay Description:Inhibition of PI4K betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase alpha(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI4K alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346968(CHEMBL1795882)
Affinity DataEC50:  10nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346969(CHEMBL1795883)
Affinity DataEC50:  10nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346970(CHEMBL1795884)
Affinity DataEC50:  1nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346971(CHEMBL1795885)
Affinity DataEC50:  150nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346972(CHEMBL1795886)
Affinity DataEC50:  150nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346973(CHEMBL1795887)
Affinity DataEC50:  25nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346974(CHEMBL1795888)
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346975(CHEMBL1795889)
Affinity DataEC50:  50nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346964(CHEMBL1795878)
Affinity DataEC50:  30nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346963(CHEMBL1795877)
Affinity DataEC50:  25nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346962(CHEMBL1795876)
Affinity DataEC50:  15nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346961(CHEMBL1795875)
Affinity DataEC50:  5nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346965(CHEMBL1795879)
Affinity DataEC50:  20nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346966(CHEMBL1795880)
Affinity DataEC50:  200nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Mus musculus (Mouse))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50346967(CHEMBL1795881)
Affinity DataEC50:  25nMAssay Description:Inhibition of mTOR-dependent S6K phosphorylation at T389 residue in MEF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed