Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50034098
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356991(CHEMBL1916247)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356988(CHEMBL1916245)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356990(CHEMBL1916246)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356980(CHEMBL1916237)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356987(CHEMBL1916244)
Affinity DataIC50:  42nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356989(CHEMBL1914477)
Affinity DataIC50:  54nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356995(CHEMBL1916251)
Affinity DataIC50:  59nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356992(CHEMBL1916248)
Affinity DataIC50:  69nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356981(CHEMBL1916238)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356986(CHEMBL1916243)
Affinity DataIC50:  75nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356985(CHEMBL1916242)
Affinity DataIC50:  82nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356996(CHEMBL1916252)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356982(CHEMBL1916239)
Affinity DataIC50:  126nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356994(CHEMBL1916250)
Affinity DataIC50:  136nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356993(CHEMBL1916249)
Affinity DataIC50:  136nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356999(CHEMBL1916412)
Affinity DataIC50:  144nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356983(CHEMBL1916240)
Affinity DataIC50:  161nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356997(CHEMBL1916253)
Affinity DataIC50:  163nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356998(CHEMBL1916254)
Affinity DataIC50:  174nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356979(CHEMBL1916236)
Affinity DataIC50:  175nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50356984(CHEMBL1916241)
Affinity DataIC50:  519nMAssay Description:Antagonist activity at human AR overexpressed in human LNCAP cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed