TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.590nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: >1nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: >1nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Homo sapiens (Human))
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Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity to EBPMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 209nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 211nMAssay Description:Binding affinity to EBPMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 233nMAssay Description:Binding affinity to EBPMore data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 368nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 372nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 419nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 455nMAssay Description:Binding affinity to EBPMore data for this Ligand-Target Pair
Affinity DataKi: 456nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 481nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 605nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 918nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair