Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50034500
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363434(CHEMBL1944782)
Affinity DataEC50:  210nMAssay Description:Partial agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363435(CHEMBL1944783)
Affinity DataEC50:  200nMAssay Description:Partial agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363436(CHEMBL1945212)
Affinity DataEC50:  680nMAssay Description:Partial agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363437(CHEMBL1945213)
Affinity DataEC50:  130nMAssay Description:Partial agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363438(CHEMBL1945214)
Affinity DataEC50:  94nMAssay Description:Partial agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363439(CHEMBL1945215)
Affinity DataEC50:  240nMAssay Description:Partial agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363445(CHEMBL1945221)
Affinity DataEC50:  67nMAssay Description:Agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363441(CHEMBL1945217)
Affinity DataEC50: >1.00E+3nMAssay Description:Partial agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363442(CHEMBL1945218)
Affinity DataEC50:  130nMAssay Description:Partial agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363443(CHEMBL1945219)
Affinity DataEC50:  320nMAssay Description:Agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363444(CHEMBL1945220)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363440(CHEMBL1945216)
Affinity DataEC50:  880nMAssay Description:Partial agonist activity at human PPARgamma expressed in MG-63 cells by reporter gene-based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed