TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Affinity DataKi: 4.50E+4nMAssay Description:Negative allosteric modulation at M2 receptor by AS-MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Competitive inhibition of Aurora A by DEL methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of SRC by DEL methodMore data for this Ligand-Target Pair
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Affinity DataKd: 1.17E+4nMAssay Description:Binding affinity to ERG by surface plasmon resonanceMore data for this Ligand-Target Pair
TargetETS translocation variant 1(Homo sapiens (Human))
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Affinity DataKd: 1.74E+4nMAssay Description:Binding affinity to ETV1 by surface plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataKd: 930nMAssay Description:Displacement of BakBH3 from Bcl-xL by DEL methodMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Affinity DataKd: 1.60E+4nMAssay Description:Binding affinity to JNK1 allosteric site by AS-MS analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Affinity DataKd: 700nMAssay Description:Orthosteric antagonist activity at M2 receptor by AS-MS analysisMore data for this Ligand-Target Pair
Affinity DataKd: 9.48E+3nMAssay Description:Inhibition of interaction of EWS-Fli1 to GST-tagged RNA Helicase A (647-1075) by surface plasmon resonanceMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Affinity DataKd: 4.80E+3nMAssay Description:Displacement of fluorescein-labeled p53 peptide from HDM2 by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Broad Institute Of Harvard And Mit
Curated by ChEMBL
Affinity DataKd: 80nMAssay Description:Displacement of fluorescein-labeled p53 peptide from HDM2 by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Antagonist activity at pirin by ITC assayMore data for this Ligand-Target Pair