Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50040853
TargetHistamine H3 receptor(Homo sapiens (Human))
Eth Zurich (Swiss Federal Institute Of Technology)

Curated by ChEMBL
LigandPNGBDBM50159110(1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piper...)
Affinity DataKi:  0.575nMAssay Description:Binding affinity to human recombinant histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataKi:  0.654nMAssay Description:Binding affinity to rat cerebral cortex histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)

Curated by ChEMBL
LigandPNGBDBM50159110(1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piper...)
Affinity DataKi:  1.26nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)

Curated by ChEMBL
LigandPNGBDBM50278350(4-fluoro-1-(4-(3-(piperidin-1-yl)propoxy)benzyl)pi...)
Affinity DataKd: >3.00E+3nMAssay Description:Binding affinity to rat histamine H3 receptor low affinity site after 1 hr by Schard plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)

Curated by ChEMBL
LigandPNGBDBM50278350(4-fluoro-1-(4-(3-(piperidin-1-yl)propoxy)benzyl)pi...)
Affinity DataKd:  0.340nMAssay Description:Binding affinity to rat brain histamine H3 receptor after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed