Affinity DataKi: 7nMAssay Description:Inhibition of CYP3A4 activity in human liver microsomes using midazolam as a substrate by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of CYP3A4 activity in human liver microsomes using nifedipine as a substrate by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Inhibition of CYP3A4 activity in human liver microsomes using testosterone as a substrate by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.80E+4nMAssay Description:Inhibition of CYP3A4 activity in human liver microsomes using midazolam as a substrate by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.87E+5nMAssay Description:Inhibition of CYP3A4 activity in human liver microsomes using testosterone as a substrate by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.03E+5nMAssay Description:Inhibition of CYP3A4 activity in human liver microsomes using nifedipine as a substrate by LC/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80nMAssay Description:Inhibition of CYP3A4 activity in human liver microsomes assessed as dibenzo fluuorescene oxidation up to 40 uMMore data for this Ligand-Target Pair
Affinity DataEC50: 0.300nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.5nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.10nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.80nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0950nMAssay Description:Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assayMore data for this Ligand-Target Pair