BindingDB PrimarySearch_ki

Found 107 Enz. Inhib. hit(s) with all data for entry = 50005570

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50039251((R)-1-(4,4-bis(3-methylthiophen-2-yl)but-3-enyl)pi...)

Ki: 39nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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3D Structure (crystal)

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492908(CHEMBL2414190)

Ki: 9.12E+3nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492912(CHEMBL2414193)

Ki: 1.15E+4nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50039246((S)-1-(2-(tris(4-methoxyphenyl)methoxy)ethyl)piper...)

Ki: 2.75E+4nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492911(CHEMBL2414173)

Ki: 4.27E+4nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492907(CHEMBL2414194)

Ki: 4.37E+4nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492893(CHEMBL2414186)

Ki: 4.68E+4nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492894(CHEMBL2414189)

Ki: 5.13E+4nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492889(CHEMBL2414187)

Ki: 5.62E+4nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492892(CHEMBL2414192)

Ki: 7.59E+4nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492895(CHEMBL2414184)

Ki: 8.13E+4nMAssay Description:Binding affinity to mouse GAT1 stably transfected in HEK293 cells by NO-711 binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50039251((R)-1-(4,4-bis(3-methylthiophen-2-yl)but-3-enyl)pi...)

IC50: 132nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed PDB

3D Structure (crystal)

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492898(CHEMBL2414176)

IC50: 7.24E+3nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492888(CHEMBL2414171)

IC50: 7.76E+3nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492890(CHEMBL2414177)

IC50: 9.55E+3nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492912(CHEMBL2414193)

IC50: 9.77E+3nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492899(CHEMBL2414175)

IC50: 1.05E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492889(CHEMBL2414187)

IC50: 1.10E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492913(CHEMBL2414178)

IC50: 1.12E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492897(CHEMBL2414179)

IC50: 1.17E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492898(CHEMBL2414176)

IC50: 1.26E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492915(CHEMBL2414182)

IC50: 1.32E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492890(CHEMBL2414177)

IC50: 1.32E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492902(CHEMBL2414078)

IC50: 1.32E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492899(CHEMBL2414175)

IC50: 1.35E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492897(CHEMBL2414179)

IC50: 1.45E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492889(CHEMBL2414187)

IC50: 1.48E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492908(CHEMBL2414190)

IC50: 1.48E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492911(CHEMBL2414173)

IC50: 1.62E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492896(CHEMBL2414181)

IC50: 1.62E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492912(CHEMBL2414193)

IC50: 1.66E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492894(CHEMBL2414189)

IC50: 1.70E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492917(CHEMBL2414081)

IC50: 1.82E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492893(CHEMBL2414186)

IC50: 1.82E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492898(CHEMBL2414176)

IC50: 1.91E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492892(CHEMBL2414192)

IC50: 1.95E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492901(CHEMBL2414079)

IC50: 1.95E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492895(CHEMBL2414184)

IC50: 2.00E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492913(CHEMBL2414178)

IC50: 2.14E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492893(CHEMBL2414186)

IC50: 2.19E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492913(CHEMBL2414178)

IC50: 2.19E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492888(CHEMBL2414171)

IC50: 2.19E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492897(CHEMBL2414179)

IC50: 2.24E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492915(CHEMBL2414182)

IC50: 2.29E+4nMAssay Description:Inhibition of mouse GAT2-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492887(CHEMBL2414188)

IC50: 2.29E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492889(CHEMBL2414187)

IC50: 2.34E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mus musculus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492894(CHEMBL2414189)

IC50: 2.34E+4nMAssay Description:Inhibition of mouse GAT3-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492890(CHEMBL2414177)

IC50: 2.34E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492914(CHEMBL2414080)

IC50: 2.40E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Jagiellonian University Medical College

Curated by ChEMBL

PNG

BDBM50492900(CHEMBL2414167)

IC50: 2.40E+4nMAssay Description:Inhibition of mouse GAT1-mediated [3H]GABA uptake stably transfected in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Details Article PubMed

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