Compile Data Set for Download or QSAR
maximum 50k data
Found 41 Enz. Inhib. hit(s) with all data for entry = 50005592
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493039(CHEMBL2418733)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493034(CHEMBL2418571)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493036(CHEMBL2418572)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493037(CHEMBL2418734)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493038(CHEMBL2418732)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493032(CHEMBL2418729)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493041(CHEMBL2418730)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493035(CHEMBL2418737)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493039(CHEMBL2418733)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493031(CHEMBL2418736)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493033(CHEMBL2418731)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493034(CHEMBL2418571)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493040(CHEMBL2418735)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493038(CHEMBL2418732)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493036(CHEMBL2418572)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493037(CHEMBL2418734)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493041(CHEMBL2418730)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493037(CHEMBL2418734)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493039(CHEMBL2418733)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493036(CHEMBL2418572)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493035(CHEMBL2418737)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493033(CHEMBL2418731)
Affinity DataKi:  136nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493034(CHEMBL2418571)
Affinity DataKi:  139nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493040(CHEMBL2418735)
Affinity DataKi:  198nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493041(CHEMBL2418730)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  299nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493032(CHEMBL2418729)
Affinity DataKi:  302nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493038(CHEMBL2418732)
Affinity DataKi:  318nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493033(CHEMBL2418731)
Affinity DataKi:  583nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  605nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493032(CHEMBL2418729)
Affinity DataKi:  721nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493035(CHEMBL2418737)
Affinity DataKi:  876nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493031(CHEMBL2418736)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493031(CHEMBL2418736)
Affinity DataKi:  1.96E+3nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKi:  2.37E+3nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50493040(CHEMBL2418735)
Affinity DataKi:  3.54E+3nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKi:  1.25E+4nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed