Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50005581
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493002(CHEMBL2413795)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain homogenates after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493000(CHEMBL2413878)
Affinity DataKi:  19nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain homogenates after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50109389(1-Phenethyl-piperidine | 1-phenethylpiperidine | C...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain homogenates after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492998(CHEMBL2413796)
Affinity DataKi:  59nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain homogenates after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493001(CHEMBL2413877)
Affinity DataKi:  84nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain homogenates after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492997(CHEMBL2413876)
Affinity DataKi:  120nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain homogenates after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492999(CHEMBL2413879)
Affinity DataKi:  790nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain homogenates after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493001(CHEMBL2413877)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492999(CHEMBL2413879)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493002(CHEMBL2413795)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492999(CHEMBL2413879)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492998(CHEMBL2413796)
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492999(CHEMBL2413879)
Affinity DataKi:  6.20E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493000(CHEMBL2413878)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492998(CHEMBL2413796)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493000(CHEMBL2413878)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493002(CHEMBL2413795)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492997(CHEMBL2413876)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492997(CHEMBL2413876)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492997(CHEMBL2413876)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493000(CHEMBL2413878)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50492998(CHEMBL2413796)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493002(CHEMBL2413795)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493001(CHEMBL2413877)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50493001(CHEMBL2413877)
Affinity DataKi:  2.10E+4nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed