TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human TNKS1 after 1 to 2 hrs by fluorescence polarization methodMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human TNKS1 after 1 to 2 hrs by fluorescence polarization methodMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human TNKS2 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human TNKS2 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human TNKS1 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human TNKS1 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of human TNKS2 after 1 to 2 hrs by fluorescence polarization methodMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of human TNKS2 after 1 to 2 hrs by fluorescence polarization methodMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human TNKS2 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Therachem Research Medilab (India)
Curated by ChEMBL
Therachem Research Medilab (India)
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:Inhibition of human TNKS1 incubated for 30 mins prior to substrate addition measured after 2 hrs by HTRF methodMore data for this Ligand-Target Pair