Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50046007
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50090908(CHEBI:67291 | CHEMBL1774404)
Affinity DataIC50:  3.00E+3nMAssay Description:Activation of GSK-3beta in HEK293 cells assessed as suppression of TCF/beta-catenin transcriptional activity after 24 hrs by SuperTOPFlash reporter g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50090907(CHEBI:66041 | CHEMBL444160)
Affinity DataIC50:  6.80E+3nMAssay Description:Activation of GSK-3beta in HEK293 cells assessed as suppression of TCF/beta-catenin transcriptional activity after 24 hrs by SuperTOPFlash reporter g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50090909(CHEMBL3120496)
Affinity DataIC50:  1.16E+4nMAssay Description:Activation of GSK-3beta in HEK293 cells assessed as suppression of TCF/beta-catenin transcriptional activity after 24 hrs by SuperTOPFlash reporter g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed