Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50047232
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155330(CHEMBL3781890)
Affinity DataIC50:  650nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155326(CHEMBL3780463)
Affinity DataIC50:  680nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155332(CHEMBL3781465)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155329(CHEMBL3779912)
Affinity DataIC50:  820nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155324(CHEMBL3780894)
Affinity DataIC50:  850nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155328(CHEMBL3781727)
Affinity DataIC50:  4.50E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155325(CHEMBL3780991)
Affinity DataIC50:  4.60E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155323(CHEMBL3781370)
Affinity DataIC50:  6.86E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155331(CHEMBL3781952)
Affinity DataIC50:  7.65E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155448(CHEMBL3781901)
Affinity DataIC50:  8.80E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandPNGBDBM50155327(CHEMBL3781940)
Affinity DataIC50:  1.08E+5nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed