Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50048814
LigandPNGBDBM94503(2-hydroxypropane-1,2,3-tricarboxylic acid;N-[4-(me...)
Affinity DataKi:  0.0200nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  2.20nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
LigandPNGBDBM50228269(CHEMBL178035)
Affinity DataKi:  3.5nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2 sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228255(CHEMBL362439)
Affinity DataKi:  7.70nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM83450(ALFENTANIL | Alfentanil hydrochloride | MLS0023206...)
Affinity DataKi:  8.20nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2 sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228260(CHEMBL367286)
Affinity DataKi:  8.20nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228221(CHEMBL366899)
Affinity DataKi:  9.10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228224(CHEMBL367667)
Affinity DataKi:  10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228217(CHEMBL174694)
Affinity DataKi:  10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228259(CHEMBL426034)
Affinity DataKi:  12nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228219(CHEMBL178847)
Affinity DataKi:  14nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228251(CHEMBL176438)
Affinity DataKi:  14nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228218(CHEMBL368487)
Affinity DataKi:  24nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228231(CHEMBL174828)
Affinity DataKi:  26nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228225(CHEMBL174758)
Affinity DataKi:  27nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228230(CHEMBL174947)
Affinity DataKi:  30nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228264(CHEMBL367661)
Affinity DataKi:  30nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228253(CHEMBL367968)
Affinity DataKi:  41nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228256(CHEMBL369412)
Affinity DataKi:  49nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228226(CHEMBL172032)
Affinity DataKi:  56nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228263(CHEMBL175126)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228257(CHEMBL172703)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228258(CHEMBL172717)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228223(CHEMBL369448)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228222(CHEMBL175148)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228250(CHEMBL369455)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228254(CHEMBL172910)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228262(CHEMBL172531)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228252(CHEMBL435340)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228268(CHEMBL173971)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228228(CHEMBL366436)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228270(CHEMBL178434)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228227(CHEMBL174962)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228265(CHEMBL263783)
Affinity DataKi: >100nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228267(CHEMBL177046)
Affinity DataKi: >100nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228229(CHEMBL174834)
Affinity DataKi: >100nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228266(CHEMBL369871)
Affinity DataKi: >100nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228220(CHEMBL174926)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228261(CHEMBL176618)
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed